V. González-Ruiz; M. Staderini; M. Bartolini; V. Andrisano; M. L. Bolognesi; N. Cabezas; J. C. Menéndez; A. I. Olives; M. A. Martína, XV International Symposium on Luminescence Spectrometry - Biophysical and Analytical Aspects, Extended Abstracts, 19-22 June 2012, Barcelona,Spain - (ISLS 2012), «LUMINESCENCE», 2012, 27, pp. 534 - 572 [Abstract]
S. Rizzo; A. Tarozzi; M. Bartolini; G. Da Costa; A. Bisi; S. Gobbi; F. Belluti; A. Ligresti; M. Allarà; J-P. Monti; V. Andrisano; V. Di Marzo; P. Hrelia; A. Rampa, 2-Arylbenzofuran-based molecules as multipotent Alzheimer's disease modifying agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2012, 58, pp. 519 - 532 [Scientific article]
F. Belluti; M. Bartolini; G. Bottegoni; A. Bisi; A. Cavalli; V. Andrisano; A. Rampa, Benzophenone-based derivatives: A novel series of potent and selective dual inhibitors of acetylcholinesterase and acetylcholinesterase-induced
beta-amyloid aggregation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 1682 - 1693 [Scientific article]
F. Mancini; A. De Simone; V. Andrisano, Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors., «ANALYTICAL AND BIOANALYTICAL CHEMISTRY», 2011, 400, pp. 1979 - 1996 [Scientific article]
Bartolini M.; Pistolozzi M.; Andrisano V.; Egea J.; Lopez M.G.; Iriepa I.; Moraleda I.; Galvez E.; Marco-Contelles J.; Samadi A., Chemical and Pharmacological Studies on Enantiomerically Pure p-Methoxytacripyrines, Promising Multi-Target-Directed Ligands for the Treatment of Alzheimer's Disease, «CHEMMEDCHEM», 2011, 6, pp. 1990 - 1997 [Scientific article]
A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre, Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment, in: Atti del XXIV Congresso Nazionale della Società Chimica Italiana, LECCE, 2011 Università del Salento – Coordinamento SIBA-, 2011, pp. 434 - 435 (atti di: XXIV Congresso Nazionale della Società Chimica Italiana, Lecce, 11-16 settembre 2011) [Abstract]
M. Rosini; E. Simoni; M. Bartolini; A. Tarozzi; R. Matera; A. Milelli; P. Hrelia; V. Andrisano; M.L. Bolognesi; C. Melchiorre, Exploiting the lipoic acid structure in the search for novel multitarget ligands against Alzheimer's disease., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 5435 - 5442 [Scientific article]
M. Bartolini; M. Naldi; J. Fiori; F. Valle; F. Biscarini; D.V. Nicolau; V. Andrisano, Kinetic characterization of amyloid-beta 1-42 aggregation with a multimethodological approach., «ANALYTICAL BIOCHEMISTRY», 2011, 414, pp. 215 - 225 [Scientific article]
S. Rizzo; A. Bisi; M. Bartolini; F. Mancini; F. Belluti; S. Gobbi; V. Andrisano; A. Rampa, Multi-target strategy to address Alzheimer’s disease: Design, synthesis and biological evaluation of new tacrine-based dimers, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 4336 - 4343 [Scientific article]
Bolognesi M.L.; Bartolini M. ; Tarozzi A.; Morroni F. ; Lizzi F. ; Milelli A. ; Minarini A. ; Rosini M.; Hrelia P.; Andrisano V.; Melchiorre C., Multitargeted drugs discovery: Balancing anti-amyloid and anticholinesterase capacity in a single chemical entity, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2011, 21, pp. 2655 - 2658 [Scientific article]
Chiriano G.; Sartini A.; Mancini F.; Andrisano V.; Bolognesi M. L.; Roberti M.; Recanatini M.; Carloni P.; Cavalli A., Sequential Virtual Screening Approach to the
Identification of Small Organic Molecules as
Potential BACE-1 Inhibitors, «CHEMICAL BIOLOGY & DRUG DESIGN», 2011, 77, pp. 268 - 271 [Scientific article]
Martins C.; Carreiras M. C.; Leon R.; de Los Rios C.; Bartolini M.; Andrisano V.; Iriepa I.; Moraleda I.; Galvez E.; Garcia M.; Egea J.; Samadi A.; Chioua M.; Marco-Contelles J., Synthesis and biological assessment of diversely substituted furo[2,3-b]quinolin-4-amine and pyrrolo[2,3-b]quinolin-4-amine derivatives, as novel tacrine analogues, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 6119 - 6130 [Scientific article]
Bolognesi ML; Chiriano G; Bartolini M; Mancini F; Bottegoni G; Maestri V; Czvitkovich S; Windisch M; Cavalli A; Minarini A; Rosini M; Tumiatti V; Andrisano V; Melchiorre C., Synthesis of Monomeric Derivatives To Probe Memoquin's Bivalent Interactions, «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 8299 - 82304 [Scientific article]
Angela De Simone; F. Mancini; C. Bertucci; V. Andrisano, A multi-approach study for BACE-1 inhibitors characterization., in: Nuove Prospettive in Chimica Farmaceutica 4, 2010, pp. 5 - 5 (atti di: NPCF4, Cagliari, 6-7 Maggio 2010) [Contribution to conference proceedings]
Bartolini M.; Naldi M.; Fiori J.; Valle F.; Biscarini F.; Nicolau D.V.; Andrisano V., A MULTI-METHODOLOGICAL APPROACH FOR BETA-AMYLOID AGGREGATION AND INHIBITION STUDIES, in: XX National Meeting on Medicinal Chemistry - Book of Abstracts, PADOVA, CLEUP sc, 2010, pp. 74 - 74 (atti di: XX National Meeting on Medicinal Chemistry, Abano Terme, Padova, September 12-16, 2010) [Abstract]