M. Bartolini; M. Naldi; D.V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van den Heuvel; V. Andrisano, ACETYLCHOLINESTERASE-BASED ANALYTICAL TOOLS FOR
DRUG SCREENING, in: Vth Conversatory on Medicinal Chemistry, LUBLIN, bestprint, 2012, pp. L-5 - L-5 (atti di: Vth Conversatory on Medicinal Chemistry - Book of Abstract, Lublin, 13-15 September 2012) [Abstract]
Naldi M.; Fiori J.; Pistolozzi M.; Drake A.F.; Bertucci C.; Wu R.; Mlynarczyk K.; Filipek S.; De Simone A.; Andrisano V., Amyloid beta-Peptide 25-35 Self Assembly and Its Inhibition: A Model Undecapeptide System to Gain Atomistic and Secondary Structure Details of the Alzheimer's Disease Process and Treatment, «ACS CHEMICAL NEUROSCIENCE», 2012, 3, pp. 952 - 962 [Scientific article]
Chlebek, Jakub; De Simone, Angela; Mancini, Francesca; Andrisano, Vincenza, An immobilized enzyme reactor based on human recombinant betasecretase (hrBACE-1-IMER) for the fast processing of substrates and screening of inhibitors, in: 21st National Meeting on Medicinal Chemistry NMMC 2012, 2012(atti di: 21st National Meeting on Medicinal Chemistry NMMC 2012, Palermo, 17-20 Luglio) [Poster]
Bartolini M.; Andrisano V, CHOLINESTERASE INHIBITION AS STARTING POINT FOR A MORE EFFECTIVE TREATMENT OF ALZHEIMER’S DISEASE, in: SINS 2012 - XIV Congress of the Italian Society for Neuroscience - 1st joint meeting with the Israel Society for Neuroscience - Program and abstract book, CATANIA, s.n, 2012, pp. 110 - 110 (atti di: SINS 2012 - XIV Congress of the Italian Society for Neuroscience - 1st joint meeting with the Israel Society for Neuroscience, Monastero dei Benedettini, Catania Italy, April 19th - 22nd, 2012) [Abstract]
De Simone, A; Mancini, F; Belluti, F; Bartolini, M; Bottegoni, G.; Rampa, A.; Cavalli, A.; Andrisano, V., Curcumin derivatives as beta-secretase (BACE1) inhibitors., in: Nuove Prospettive in Chimica Farmaceutica 6, 2012(atti di: Nuove Prospettive in Chimica Farmaceutica 6, Riccione, 11-13 Aprile) [Poster]
Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S., Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment., «NEUROPHARMACOLOGY», 2012, 62, pp. 997 - 1003 [Scientific article]
J. Fiori; M. Naldi; M. Bartolini; V. Andrisano, Disclosure of a fundamental clue for the elucidation of the myricetin mechanism of action as amyloid aggregation inhibitor by mass spectrometry, «ELECTROPHORESIS», 2012, 33, pp. 1 - 7 [Scientific article]
Galdeano C.; Viayna E.; Sola I.; Formosa X.; Camps P. Badia A.; Clos M.V.; Relat J.; Ratia M.; Bartolini M.; Mancini F.; Andrisano V.; Salmona M.; Minguillon C.; Gonzalez-Munoz G. C.; Rodriguez-Franco M. I.; Bidon-Chanal A.; Luque F. J.; Munoz-Torrero D., Huprine-tacrine heterodimers as anti-amyloidogenic compounds of potential interest against Alzheimer's and prion diseases, «JOURNAL OF MEDICINAL CHEMISTRY», 2012, 55, pp. 661 - 669 [Scientific article]
Kacker, Puneet; De Simone, Angela; Masetti, Matteo; Bottegoni, Giovanni; Andrisano, Vincenza; Cavalli, Andrea, Identification of Novel BACE-1 Inhibitors through an Advanced Structure-Based Virtual Screening Protocol., in: Structural & Computational Chemistry Congress, 2012(atti di: Structural & Computational Chemistry Congress, Munich, Germany, 13-14 March 2012) [Poster]
Parolin C; Calonghi N; Presta E; Boga C; Caruana P; Naldi M; Andrisano V; Masotti L; Sartor G., Mechanism and stereoselectivity of HDAC I inhibition by (R)-9-hydroxystearic acid in colon cancer., «BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS», 2012, 10, pp. 1334 - 1340 [Scientific article]
Samadi A.; de los Ríos C.; Bolea I.; Chioua M.; Iriepa I.; Moraleda I.; Bartolini M.; Andrisano V.; Gálvez E.; Valderas C.; Unzeta M.; Marco-Contelles J., Multipotent MAO and cholinesterase inhibitors for the treatment of Alzheimer's disease: synthesis, pharmacological analysis and molecular modeling of heterocyclic substituted alkyl and cycloalkyl propargyl amine., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2012, 52, pp. 251 - 262 [Scientific article]
Cosconati S.; Marinelli L.; Di Leva F.S.; La Pietra V.; De Simone A.; Mancini F.; Andrisano V.; Novellino E.; Goodsell D.S.; Olson A.J., Protein Flexibility in Virtual Screening: The BACE-1 Case Study, «JOURNAL OF CHEMICAL INFORMATION AND MODELING», 2012, 52, pp. 2697 - 2704 [Scientific article]
Simoni E.; Rosini M.; Bartolini M.; Andrisano V.; Soriano E.; Marco-Contelles J.; Melchiorre C.; Bolognesi M.L., Rational design of dimebon bivalent ligands against Alzheimer’s disease, in: Libro degli abstracts, s.l, s.n, 2012, pp. 38 - 38 (atti di: NPCF6-Nuove prospettive in chimica farmaceutica- 6°Meeting, Riccione, 15-17 aprile 2012) [Abstract]
A. Rampa; M. Bartolini; A. Bisi; F. Belluti; S. Gobbi; V. Andrisano; A. Ligresti; V. Di Marzo, The first dual ChE/FAAH inhibitors: new perspectives for
Alzheimer's disease?, «ACS MEDICINAL CHEMISTRY LETTERS», 2012, 3, pp. 182 - 186 [Scientific article]
Pulawski W; Ghoshdastider U; Andrisano V; Filipek S, Ubiquitous amyloids, «APPLIED BIOCHEMISTRY AND BIOTECHNOLOGY», 2012, 166, pp. 1626 - 1643 [Scientific article]
