vai alle Pubblicazioni
Publications prior to 2004
Pubblicazioni antecedenti il 2004
1)
A. Andreani, A. Locatelli, A. Leoni, M. Rambaldi, R. Morigi, R.
Bossa, M. Chiericozzi, A. Fraccari, I. Galatulas.
Synthesis and potential coanthracyclinic activity of
substituted
3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones. Eur. J. Med.
Chem. 32, 919-924
(1997).
2)
A. Andreani, A. Leoni, R. Morigi, R. Bossa, M.
Chiericozzi, I. Galatulas.
In vivo cardiotonic activity of aryl- and
pyridyl- substituted fused imidazoles. Arzneim.-Forsch./Drug Res. 48 (I), 3,
232-235 (1998).
3)
A. Andreani, A. Locatelli,
R. Morigi, A. Leoni, R. Bossa, M. Chiericozzi, I.
Galatulas.
In vivo cardiotonic activity of
pyridylmethylene-2-indolinones. Arzneim.-Forsch./Drug Res.
48 (II), 7, 727-729 (1998).
4)
A. Andreani, A. Leoni, A.
Locatelli, R. Morigi, M. Chiericozzi, A. Fraccari, I.
Galatulas.
Potential coanthracyclinic activity of
pyridylmethylene-2-indolinones. Anticancer
Res. 18, 3407-3410
(1998).
5)
A. Andreani, A. Locatelli, A. Leoni, R. Morigi, M. Chiericozzi, A.
Fraccari, I. Galatulas, G. Salvatore.
Synthesis and potential coanthracyclinic activity of
pyridylmethylene and indolylmethylene lactams. Eur. J. Med.
Chem. 33, 905-909,
(1998).
6)
A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, J.C.
Gehret, S. Traniello, A. Cariani, S. Spisani.
Ring-opened analogs of indomethacin affecting human
neutrophil functions. Collect. Czech.
Chem. Commun. 64, 299-312,
(1999).
7)
A. Andreani, M. Rambaldi, A. Leoni, R. Morigi, A. Locatelli, G.
Giorgi, G. Lenaz, A. Ghelli, M. Degli Esposti.
6-Thienyl and 6-phenylimidazo[2,1-b]thiazoles as
inhibitors of mitochondrial NADH dehydrogenase. Eur. J. Med.
Chem. 34, 883-889,
(1999).
8)
A. Andreani, A. Leoni, A.
Locatelli, R. Morigi, M. Rambaldi, C. Pietra, G.
Villetti.
4-Aminopyridine derivatives with antiamnesic
activity. Eur. J. Med.
Chem. 35, 77-82,
(2000).
9)
A. Andreani, M. Rambaldi, A.
Leoni, A. Locatelli, R. Morigi, S. Traniello, A. Cariani, O.
Rizzuti, S. Spisani.
6-(Hydroxyphenyl)imidazo[2,1-b]thiazoles as potential
antiinflammatory agents: effects on human neutrophil
functions. Collect. Czech.
Chem. Commun. 65, 267-279,
(2000).
10)
A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, W.A.
Simon, J. Senn-Bilfinger.
Synthesis and antisecretory activity of 6-substituted
5-cyanomethylimidazo[2,1-b]thiazoles and
2,6-dimethyl-5-hydroxymethylimidazo[2,1-b][1,3,4]thiadiazole.
Arzneim.-Forsch./Drug
Res. 50 (I), 6,
550-553, (2000).
11)
A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, M.
Recanatini, V. Garaliene.
Potential antitumor agents. Part 29. Synthesis and
potential coanthracyclinic activity of imidazo[2,1-b]thiazole
guanylhydrazones. Bioorg. Med.
Chem. 8, 2359-2366,
(2000).
12)
A. Andreani, A. Cavalli, M. Granaiola, A. Leoni, A. Locatelli, R.
Morigi, M. Rambaldi, M. Recanatini, M. Garnier, L.
Meijer.
Imidazo[2,1-b]thiazolylmethylene- and
indolylmethylene-2-indolinones: a new class of cyclin-dependent
kinase inhibitors. Design, synthesis and CDK1/cyclin B inhibition.
Anti-Cancer Drug
Design. 15, 447-452,
(2000).
13)
A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M.
Rambaldi.
Synthesis and antitubercular activity of
imidazo[2,1-b]thiazoles. Eur. J. Med.
Chem. 36, 743-746
(2001).
14)
A. Andreani, A. Cavalli, M. Granaiola, M. Guardigli, A. Leoni, A.
Locatelli, R. Morigi, M. Rambaldi, M. Recanatini, A.
Roda.
Synthesis and screening for antiacetylcholinesterase
activity of (1-benzil-4-oxopiperidin-3-ylidene)methylindoles and
–pyrroles related to donezepil. J. Med.
Chem. 44, 4011-4014
(2001).
15)
A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M.
Rambaldi, G. Giorgi, L. Salvini, V. Garaliene.
Synthesis and antitumor activity of substituted
3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones. Anti-Cancer
Drug Design 16, 167-174
(2001).
16)
A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M.
Rambaldi, V. Garaliene.
Synthesis and antitumor activity of 1,5,6-substituted
E-3-(2-chloro-3-indolylmethylene)-1,3-dihydroindol-2-ones.
J. Med.
Chem. 45, 2666-2669
(2002).
17)
A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R.
Morigi, M. Rambaldi, G. Giorgi, L. Salvini.
Cancer fighting cancer: synthesis of the new
heterocyclic system diimidazo[1,2-a:1,2-c]pyrimidine. Arkivoc (XI) 32-38
(2002) (Issue in Honor of Prof. Domenico
Spinelli)
http://www.arkat-usa.org/ark/journal/2002/Spinelli/Spinelli_index.htm