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Eleonora Diamanti

Ricercatrice a tempo determinato tipo a) (junior)

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHEM-07/A Chimica farmaceutica

Pubblicazioni

Braun-Cornejo, Maria; Platteschorre, Mitchell; de Vries, Vincent; Bravo, Patricia; Sonawane, Vidhisha; Hamed, Mostafa M.; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K. H., Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity, «JACS AU», 2025, 5, pp. 1146 - 1156 [articolo]

Willocx, Daan; Diamanti, Eleonora; Hirsch, Anna K. H., Targeting IspD for Anti-infective and Herbicide Development: Exploring Its Role, Mechanism, and Structural Insights, «JOURNAL OF MEDICINAL CHEMISTRY», 2025, 68, pp. 886 - 901 [articolo]

Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fato, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura, Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases, «ACS MEDICINAL CHEMISTRY LETTERS», 2024, 15, pp. 1506 - 1515 [articolo]

Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupenthal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H., Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target, «PROTEIN SCIENCE», 2024, 33, pp. 1 - 11 [articolo]Open Access

Willocx, Daan; D'Auria, Lucia; Walsh, Danica; Scherer, Hugo; Alhayek, Alaa; Hamed, Mostafa M.; Borel, Franck; Diamanti, Eleonora; Hirsch, Anna Katharina Herta, Fragment Discovery by X‐ray Crystallographic Screening Targeting the CTP Binding Site of Pseudomonas aeruginosa IspD, «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2024, 65, pp. 1 - 6 [articolo]Open Access

Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura, Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach, «ACS INFECTIOUS DISEASES», 2024, 10, pp. 1856 - 1870 [articolo]Open Access

Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Michael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H., Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT, «CHEMICAL COMMUNICATIONS», 2024, 60, pp. 870 - 873 [articolo]

Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mostafa M.; Hirsch, Anna K.H., IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding, «STRUCTURE», 2024, 32, pp. 1 - 9 [articolo]

Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Diamanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H., Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE, «ACS OMEGA», 2024, 9, pp. 38160 - 38168 [articolo]

Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Boris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H., Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity, «JOURNAL OF MEDICINAL CHEMISTRY», 2024, 67, pp. 17070 - 17086 [articolo]Open Access

Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour, Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H., Targeting the Plasmodium falciparum IspE Enzyme, «ACS OMEGA», 2024, 9, pp. 44465 - 44473 [articolo]

Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, Julien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias, Back in Person: Frontiers in Medicinal Chemistry 2023, «CHEMMEDCHEM», 2023, 18, pp. e202300344 - 1 [articolo]Open Access

Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria, Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?, «CHEMMEDCHEM», 2023, 18, Article number: e202300422, pp. 1 - 17 [articolo]Open Access

Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H, Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors, «CHEMMEDCHEM», 2023, 18, pp. e202300346 - 1 [articolo]Open Access

Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H, Identification of inhibitors targeting the energy-coupling factor (ECF) transporters, «COMMUNICATIONS BIOLOGY», 2023, 6, pp. 1 - 8 [articolo]Open Access

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