Brevetto n. US8927533, Novel process for the synthesis of 7-chloro-4-(piperazin-1-yl)-quinoline.
Baruchello R; Simoni D; Grisolia G; Barbato G; Marchetti P; Rondanin R; Mangiola S; Giannini G; Brunetti T; Alloatti D; Gallo G; Ciacci A; Vesci L; Castorina M; Milazzo FM; Cervoni ML; Guglielmi MB; Barbarino M; Fodera R; Pisano C; Cabri W, Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90, «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 8592 - 8604 [replica/breve intervento]
Botta CB; Cabri W; Cini E; De Cesare L; Fattorusso C; Giannini G; Persico M; Petrella A; Rondinelli F; Rodriquez M; Russo A; Taddei M, Oxime Amides as a Novel Zinc Binding Group in Histone Deacetylase Inhibitors: Synthesis, Biological Activity, and Computational Evaluation, «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 2165 - 2182 [replica/breve intervento]
Santaniello M; Critelli L; Quattrociocchi G; Longo A; Cabri W, Reconstituted ocular gel for cystinosis treatment, «JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY», 2011, 21, pp. 273 - 277 [replica/breve intervento]
F. Gasparrini; W. Cabri; I. D'Acquarica; P. Simone; M. Di Iorio; M. Di Mattia; F. Giorgi; A. Mazzanti; M. Pierini; M. Quaglia; C. Villani, Stereolability of Dihydroartemisinin, an Antimalarial Life-Saving Drug: a Comprehensive Kinetic Investigation - Part II, «JOURNAL OF ORGANIC CHEMISTRY», 2011, 76, pp. 4831 - 4840 [articolo]
F. Gasparrini; W. Cabri; I. D'Acquarica; P. Simone; M. Di Iorio; M. Di Mattia; F. Giorgi; A. Mazzanti; M. Pierini; M. Quaglia; C.Villani, Stereolability of Dihydroartemisinin, an Antimalarial Life-Saving Drug: a Comprehensive Thermodynamic Investigation. Part I, «JOURNAL OF ORGANIC CHEMISTRY», 2011, 76, pp. 1751 - 1758 [articolo]
Gattinoni S; De Simone C; Dallavalle S; Fezza F; Nannei R; Battista N; Minetti P; Quattrociocchi G; Caprioli A; Borsini F; Cabri W; Penco S; Merlini L; Maccarrone M, A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2010, 20, pp. 4406 - 4411 [replica/breve intervento]
Tassoni E; Conti R; Gallo G; Vincenti S; Dell'Uomo N; Mastrofrancesco L; Ricciolini R; Cabri W; Carminati P; Giannessi F, Aminocarnitine Ureidic Derivatives as Inhibitors of Carnitine Palmitoyltransferase I, «CHEMMEDCHEM», 2010, 5, pp. 666 - 669 [replica/breve intervento]
Brevetto n. US9302998, ARYL TRIAZOLE COMPOUNDS WITH ANTITUMOURAL ACTIVITY.
Brevetto n. WO2010105930, CARBAMATE DERIVATIVES IN PARTICULAR FOR THE TREATMENT OF NEUROLOGICAL DISORDERS.
Bartoccini F; Cabri W; Celona D; Minetti P; Piersanti G; Tarzia G, Direct B-Alkyl Suzuki-Miyaura Cross-Coupling of 2-Halopurines. Practical Synthesis of ST1535, a Potent Adenosine A(2A) Receptor Antagonist, «JOURNAL OF ORGANIC CHEMISTRY», 2010, 75, pp. 5398 - 5401 [replica/breve intervento]
Gattinoni S; De Simone C; Dallavalle S; Fezza F; Nannei R; Amadio D; Minetti P; Quattrociocchi G; Caprioli A; Borsini F; Cabri W; Penco S; Merlini L; Maccarrone M, Enol Carbamates as Inhibitors of Fatty Acid Amide Hydrolase (FAAH) Endowed with High Selectivity for FAAH over the Other Targets of the Endocannabinoid System, «CHEMMEDCHEM», 2010, 5, pp. 357 - 360 [articolo]
Badaloni E; Cabri W; Ciogli A; D'Acquarica I; Deias R; Gasparrini F; Giorgi F; Kotoni D; Villani C, Extending the use of "Inverted Chirality Columns Approach" for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative, «JOURNAL OF CHROMATOGRAPHY A», 2010, 1217, pp. 1024 - 1032 [articolo]
Brevetto n. WO2011047926, NON-NATURAL MACROCYCLIC AMIDE HDAC6 INHIBITOR COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS.
Auzzas L; Larsson A; Matera R; Baraldi A; Deschenes-Simard B; Giannini G; Cabri W; Battistuzzi G; Gallo G; Ciacci A; Vesci L; Pisano C; Hanessian S, Non-Natural Macrocyclic Inhibitors of Histone Deacetylases: Design, Synthesis, and Activity, «JOURNAL OF MEDICINAL CHEMISTRY», 2010, 53, pp. 8387 - 8399 [replica/breve intervento]