Foto del docente

Vincenza Andrisano

Full Professor

Department for Life Quality Studies

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

L.Piazzi; A. Cavalli; F. Colizzi; F. Belluti; M. Bartolini; F. Mancini; M. Recanatini; V. Andrisano; A. Rampa, Multi-target-directed coumarin derivatives: hAChE and BAC1 inhibitors as potential anti-Alzheimer compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2008, 18, pp. 423 - 426 [Scientific article]

P. Camps; X. Formosa; C. Galdeano; T. Gòmez; D. Munoz-Torrero; M. Scarpellini; E. Viayna; A. Badia; M.V. Clos; A. Camins; M. Pallàs; M. Bartolini; F. Mancini; V. Andrisano; J. Estelrich; M. Lizondo; A. Bidon-Chanal; F.J. Luque, Novel Donepezil-Based Inhibitors of Acetyl- and Butyrylcholinesterase and Acetylcholinesterase-Induced Beta-Amyloid Aggregation, «JOURNAL OF MEDICINAL CHEMISTRY», 2008, 51, pp. 3588 - 3598 [Scientific article]

M. Bartolini; Nigel H. Greig; V. Andrisano, ON-LINE CHARACTERIZATION OF CHOLINESTERASE INHIBITORS BY IMMOBILIZED ENZYME REACTORS, in: PBA 2008 - 19th International Symposium on Pharmaceutical and Biomedical Analysis, s.l, Justyna Lapinska, 2008, pp. 315 - 315 (atti di: PBA 2008 - 19th International Symposium on Pharmaceutical and Biomedical Analysis, Gdansk, Poland, 8-12 Giugno 2008) [Abstract]

Coordination of a Research Project: PRIN 2007 Metodologie analitiche avanzate nelle ricerca e sviluppo di farmaci'..

S. Rizzo; A. Cavalli; L. Ceccarini; F. Belluti; A. Bisi; M. Bartolini; V. Andrisano; M. Recanatini; A. Rampa, SAR and binding mode at the h-AChE active site of pseudo-irreversible inhibitors related to Xanthostigmine, in: XIX National Meeting on Medicinal Chemistry, s.l, s.n, 2008, pp. 219 - 219 (atti di: XIX National Meeting on Medicinal Chemistry, Verona, 14-18 september 2008) [Abstract]

V. Tumiatti; A. Milelli; A. Minarini; M. Rosini; M. L. Bolognesi; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; C. Melchiorre, Structure-Activity Relationships of Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone. 4. Futher Investigation on the Inner Spacer., «JOURNAL OF MEDICINAL CHEMISTRY», 2008, 51, pp. 7308 - 7312 [Scientific article]

V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre, Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone, in: Atti del XIII Meeting Strutture eterocicliche nella ricerca farmaceutica, s.l, s.n, 2008, pp. 207 - 207 (atti di: XIII Meeting Strutture eterocicliche nella ricerca farmaceutica, Palermo, 18-21 Maggio 2008) [Abstract]

ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tumiatti; C. Melchiorre, Synthesis of monomeric derivatives to probe Memoquin bivalent interactions, in: Book of Abstracts, s.l, s.n, 2008, pp. 226 - 226 (atti di: XIX National Meeting on Medicinal Chemistry, Verona, 14-18 September 2008) [Abstract]

Petraglio G.; Bartolini M.; Branduardi D.; Andrisano V.; Recanatini M.; Gervasio F. L.; Cavalli A.; Parrinello M., The role of Li(+), Na(+), and K(+) in the ligand binding inside the human acetylcholinesterase gorge, «PROTEINS», 2008, 70, pp. 779 - 785 [Scientific article]

Cavalli A.; Bolognesi M. L.; Capsoni S.; Andrisano V.; Bartolini M.; Margotti E.; Cattaneo A.; Recanatini M.; Melchiorre C., A small molecule targeting the multifactorial nature of Alzheimer's disease, «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2007, 46, pp. 3689 - 3692 [Scientific article]

Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V., Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors., in: Frontiers in CNS and oncology medicinal chemistry-program and abstracts, s.l, s.n, 2007, pp. 51 - 52 (atti di: Frontiers in CNS and oncology medicinal chemistry, Siena (Italy), 7-9 October, 2007) [Abstract]

S. Olmo; R. Gotti; M. Naldi; V. Andrisano; N. Calonghi; V. Cavrini., CE Analysis of Basic Proteins and H4 Human Histones using a Pullulan-Coated Capillary, in: 12th Intenational Meeting on Recent Development in Pharmaceutical Analysis. RDPA 2007. Abstract Book., s.l, s.n, 2007, pp. 85 - 85 (atti di: 12th Intenational Meeting on Recent Development in Pharmaceutical Analysis. RDPA 2007., Island of Elba, Italy, September 23-26, 2007) [Abstract]

M. Bartolini; M.L. Bolognesi; A. Cavalli; C. Melchiorre; A. Rampa; M. Recanatini; V. Andrisano, Characterization of Cholinesterase inhibitors by means of immobilized enzyme reactor, in: The IXth International Meeting on Cholinesterases, Program Book, s.l, s.n, 2007, pp. 69 - 69 (atti di: IXth International Meeting on Cholinesterases, Suzhou, China, 6-10 Maggio 2007) [Contribution to conference proceedings]

Manuela Bartolini; Vanni Cavrini; Vincenza Andrisano, Characterization of reversible and pseudo-irreversible Acetylcholinesterase inhibitors by means of immobilized enzyme reactor, «JOURNAL OF CHROMATOGRAPHY A», 2007, 1144, pp. 102 - 110 [Scientific article]

L. Piazzi; F. Belluti; A. Bisi; S. Gobbi; S. Rizzo; M. Bartolini; V. Andrisano; M. Recanatini; A. Rampa, CHOLINESTERASE INHIBITORS: SAR AND ENZYME INHIBITORY ACTIVITY OF 3-[omega-(BENZYLMETHYLAMINO)ALKOXY]XANTHEN-9-ONES, «BIOORGANIC & MEDICINAL CHEMISTRY», 2007, 15, pp. 575 - 585 [Scientific article]