Bisi A.; Rampa A.; Budriesi R.; Gobbi S.; Belluti F.; Ioan P.; Valoti E.; Chiarini A.; Valenti P., Cardiovascular hybrid drugs: New benzazepinone derivatives as bradycardic agents endowed with selective β1-Non-competitive antagonism, «BIOORGANIC & MEDICINAL CHEMISTRY», 2003, 11, pp. 1353 - 1361 [Scientific article]
Budriesi R.; Cosimelli B.; Ioan P.; Lanza C.Z.; Spinelli D.; Chiarini A., Cardiovascular characterization of [1,4]thiazino[3,4-c][1,2,4]oxadiazol-1-one derivatives: Selective myocardial calcium channel modulators, «JOURNAL OF MEDICINAL CHEMISTRY», 2002, 45, pp. 3475 - 3481 [Scientific article]
Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Hucho F.; Melchiorre C., Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms, «JOURNAL OF MEDICINAL CHEMISTRY», 2002, 45, pp. 1860 - 1878 [Scientific article]
Li Y.; Popaj K.; Lochner M.; Geneste H.; Budriesi R.; Chiarini A.; Melchiorre C.; Hesse M., Analogues of polyamine alkaloids and their synthetic advantages, «IL FARMACO», 2001, 56, pp. 127 - 131 [Scientific article]
Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C., Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines, «BRITISH JOURNAL OF PHARMACOLOGY», 2001, 132, pp. 1009 - 1016 [Scientific article]Open Access
Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J., Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 4035 - 4038 [Scientific article]
Teodori E.; Dei S.; Garnier-Suillerot A.; Quidu P.; Scapecchi S.; Budriesi R., Structure-activity relationship studies on the potent multidrug resistance (MDR) modulator 2-(3,4-dimethoxyphenyl)-2-(methylethyl)-5[(anthr-9-yl) methylamino]pentanenitrile (MM 36), «MEDICINAL CHEMISTRY RESEARCH», 2001, 10, pp. 563 - 576 [Scientific article]
Dei S.; Teodori E.; Garnier-Suillerot A.; Gualtieri F.; Scapecchi S.; Budriesi R.; Chiarini A., Structure-activity relationships and optimisation of the selective MDR modulator 2-(3,4-dimethoxyphenyl)-5-(9-fluorenylamino)-2-(methylethyl) pentanenitrile and its N-methyl derivative, «BIOORGANIC & MEDICINAL CHEMISTRY», 2001, 9, pp. 2673 - 2682 [Scientific article]
Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C., Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 5212 - 5223 [Scientific article]
Teodori E.; Dei S.; Quidu P.; Budriesi R.; Chiarini A.; Garnier-Suillerot A.; Gualtieri F.; Manetti D.; Romanelli M.N.; Scapecchi S., Design, synthesis, and in vitro activity of catamphiphilic reverters of multidrug resistance: Discovery of a selective, highly efficacious chemosensitizer with potency in the nanomolar range, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 1687 - 1697 [Scientific article]
Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 4214 - 4224 [Scientific article]
Valenti P.; Rampa A.; Budriesi R.; Bisi A.; Chiarini A., Coumarin 1,4-dihydropyridine derivatives, «BIOORGANIC & MEDICINAL CHEMISTRY», 1998, 6, pp. 803 - 810 [Scientific article]
Bolognesi M.L.; Budriesi R.; Chiarini A.; Poggesi E.; Leonardi A.; Melchiorre C., Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for α1-adrenoreceptor subtypes, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4844 - 4853 [Scientific article]
Melchiorre C.; Bolognesi M.L.; Budriesi R.; Chiarini A.; Giardina D.; Minarini A.; Quaglia W.; Leonardi A., Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?, «IL FARMACO», 1998, 53, pp. 278 - 286 [Scientific article]
