Foto del docente

Marinella Roberti

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Bagnolini, G.; Balboni, B.; Schipani, F.; Gioia, D.; Veronesi, M.; De Franco, F.; Kaya, C.; Jumde, R. P.; Ortega, J. A.; Girotto, S.; Hirsch, A. K. H.; Roberti, M.; Cavalli, A., Identification of RAD51-BRCA2 Inhibitors Using N-Acylhydrazone-Based Dynamic Combinatorial Chemistry, «ACS MEDICINAL CHEMISTRY LETTERS», 2022, 13, pp. 1262 - 1269 [Scientific article]Open Access

Bagnolini, Greta; Balboni, Beatrice; Schipani, Fabrizio; Gioia, Dario; Veronesi, Marina; De Franco, Francesca; Kaya, Cansu; Jumde, Ravindra P.; Antonio Ortega, Jose; Girotto, Stefania; Hirsch, Anna K. H.; Roberti, Marinella; Cavalli, Andrea, Identification of RAD51-BRCA2 inhibitors using N-acylhydrazone-based dynamic combinatorial chemistry, in: Book of abstract, 2022, pp. 1 - 1 (atti di: HIPS Symposium 2022, Virtual, 12 May 2022) [Contribution to conference proceedings]

Previtali V., Myers S. H., Bagnolini G., Poppi L., Rinaldi F., Schipani F., Ortega J. A., De Franco F., Pellicciari R., Girotto S., Oliviero G., Walsh N., Valenti G., Tirelli N., Di Stefano G., Roberti M., Cavalli A., Insights into the activity of ARN24089, a new RAD51-BRCA2 disruptor that inhibits homologous recombination and achieves synthetic lethality in pancreatic cancer, in: ACS Spring 2022, 2022, pp. 1 - 1 (atti di: ACS Spring 2022, San Diego Convention Center, Room 16A, 20/03/2023) [Abstract]

Brusa I.; Sondo E.; Falchi F.; Pedemonte N.; Roberti M.; Cavalli A., Proteostasis Regulators in Cystic Fibrosis: Current Development and Future Perspectives, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 5212 - 5243 [Scientific article]Open Access

Schipani, Fabrizio; Manerba, Marcella; Marotta, Roberto; Poppi, Laura; Gennari, Arianna; Rinaldi, Francesco; Armirotti, Andrea; Farabegoli, Fulvia; Roberti, Marinella; Di Stefano, Giuseppina; Rocchia, Walter; Girotto, Stefania; Tirelli, Nicola; Cavalli, Andrea, The Mechanistic Understanding of RAD51 Defibrillation: A Critical Step in BRCA2-Mediated DNA Repair by Homologous Recombination, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2022, 23, Article number: 8338 , pp. 1 - 14 [Scientific article]Open Access

Bruno, F.; Castelli, G.; Vitale, F.; Catanzaro, S.; Badaco, V. V.; Roberti, M.; Colomba, C.; Cascio, A.; Tolomeo, M., Antiparasitic effect of stilbene and terphenyl compounds against trypanosoma cruzi parasites, «PHARMACEUTICALS», 2021, 14, Article number: 1199 , pp. 1 - 16 [Scientific article]Open Access

Mazzei L.; Contaldo U.; Musiani F.; Cianci M.; Bagnolini G.; Roberti M.; Ciurli S., Inhibition of Urease, a Ni-Enzyme: The Reactivity of a Key Thiol With Mono- and Di-Substituted Catechols Elucidated by Kinetic, Structural, and Theoretical Studies, «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2021, 60, pp. 6029 - 6035 [Scientific article]Open Access

Balboni, A.; Govoni, M.; Rossi, V.; Roberti, M.; Cavalli, A.; Di Stefano, G.; Manerba, M., Lactate dehydrogenase inhibition affects homologous recombination repair independently of cell metabolic asset; implications for anticancer treatment, «BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS», 2021, 1865, Article number: 129760 , pp. 1 - 10 [Scientific article]Open Access

Bagnolini, Greta; Manerba, Marcella; Balboni, Andrea; Antonio Ortega, Jose; Gioia, Dario; De Franco, Francesca; Roberti, Marinella; Cavalli, Andrea, Dihydroquinoline pyrazoline-based compound as a new RAD51-BRCA2 protein-protein disruptor to trigger synthetic lethality in pancreatic cancer, in: 1, 2020(atti di: Italian Young Medicinal Chemistry Virtual Meeting 2020, Virtual, 22-24 July 2020) [Poster]

Vetica F.; Sansone A.; Meliota C.; Batani G.; Roberti M.; Chatgilialoglu C.; Ferreri C., Free-radical-mediated formation of trans-cardiolipin isomers, analytical approaches for lipidomics and consequences of the structural organization of membranes, «BIOMOLECULES», 2020, 10, Article number: 1189 , pp. 1 - 18 [Scientific article]Open Access

Linciano P.; Cullia G.; Borsari C.; Santucci M.; Ferrari S.; Witt G.; Gul S.; Kuzikov M.; Ellinger B.; Santarem N.; Cordeiro da Silva A.; Conti P.; Bolognesi M.L.; Roberti M.; Prati F.; Bartoccini F.; Retini M.; Piersanti G.; Cavalli A.; Goldoni L.; Bertozzi S.M.; Bertozzi F.; Brambilla E.; Rizzo V.; Piomelli D.; Pinto A.; Bandiera T.; Costi M.P., Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2020, 189, Article number: 112047 , pp. N/A - N/A [Scientific article]

Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; Farabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A., Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 2588 - 2619 [Scientific article]Open Access

Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura*, A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential, «ACS CHEMICAL NEUROSCIENCE», 2019, 10, pp. 279 - 294 [Scientific article]

Camilla Marasca, Irene Brusa, Chiara Cabrelle, Michele Protti, Matteo Micucci, Laura Mercolini, Marinella Roberti, Roberta Budriesi, Maurizio Recanatini, Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources, in: Merck Young Chemists' Symposium (MYCS 2019), 2019, pp. 027 - 027 (atti di: Merck Young Chemists' Symposium (MYCS 2019), Rimini (Italia), 25-27 novembre 2019) [Contribution to conference proceedings]

Bagnolini, Greta; Balboni, Andrea; Manerba, Marcella; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Roberti, Marinella; Cavalli, Andrea, Design and synthesis of BRCA2-RAD51 disruptors to induce synthetic lethality in anticancer therapy, in: 1, 2019(atti di: WORKSHOP: I chimici per le biotecnologie, Milan, 22 February 2019) [Poster]

Latest news

At the moment no news are available.