Santino F.; Petruzzelli R.; Zhao J.; Boanini E.; Gentilucci L., Peptide bond formation using unprotected N-carboxyanhydrides under green chemistry conditions, «SUSTAINABLE CHEMISTRY AND PHARMACY», 2021, 24, Article number: 100540, pp. 1 - 8 [articolo]Open Access
Piekielna-Ciesielska, Justyna; Artali, Roberto; Azzam, Ammar A H; Lambert, David G; Kluczyk, Alicja; Gentilucci, Luca; Janecka, Anna, Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation, «MOLECULES», 2021, 26, Article number: 13, pp. 1 - 20 [articolo]Open Access
Bedini A.; Di Cesare Mannelli L.; Micheli L.; Baiula M.; Vaca G.; De Marco R.; Gentilucci L.; Ghelardini C.; Spampinato S., Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist, «FRONTIERS IN PHARMACOLOGY», 2020, 11, Article number: 188, pp. 1 - 22 [articolo]Open Access
Anselmi M.; Stavole P.; Boanini E.; Bigi A.; Juaristi E.; Gentilucci L., Green synthesis of bioactive oligopeptides promoted by recyclable nanocrystalline hydroxyapatite, «FUTURE MEDICINAL CHEMISTRY», 2020, 12, pp. 1 - 17 [articolo]Open Access
De Marco R.; Rampazzo E.; Zhao J.; Prodi L.; Paolillo M.; Picchetti P.; Gallo F.; Calonghi N.; Gentilucci L., Integrin-targeting dye-doped peg-shell/silica-core nanoparticles mimicking the proapoptotic Smac/DIABLO protein, «NANOMATERIALS», 2020, 10, Article number: 1211, pp. 1 - 13 [articolo]Open Access
Zhao J.; Santino F.; Giacomini D.; Gentilucci L., Integrin-targeting peptides for the design of functional cell-responsive biomaterials, «BIOMEDICINES», 2020, 8, Article number: 307, pp. 1 - 35 [articolo]Open Access
Stefan A.; Gentilucci L.; Piaz F.D.; D'Alessio F.; Santino F.; Hochkoeppler A., Purification from Deinococcus radiodurans of a 66 kDa ABC transporter acting on peptides containing at least 3 amino acids, «BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS», 2020, 529, pp. 869 - 875 [articolo]Open Access
Martelli G.; Baiula M.; Caligiana A.; Galletti P.; Gentilucci L.; Artali R.; Spampinato S.; Giacomini D., Could Dissecting the Molecular Framework of β-Lactam Integrin Ligands Enhance Selectivity?, «JOURNAL OF MEDICINAL CHEMISTRY», 2019, 62, pp. 10156 - 10166 [articolo]Open Access
Wtorek K.; Artali R.; Piekielna-Ciesielska J.; Koszuk J.; Kluczyk A.; Gentilucci L.; Janecka A., Endomorphin-2 analogs containing modified tyrosines: Biological and theoretical investigation of the influence on conformation and pharmacological profile, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 179, pp. 527 - 536 [articolo]
De Marco R.; Zhao J.; Greco A.; Ioannone S.; Gentilucci L., In-Peptide Synthesis of Imidazolidin-2-one Scaffolds, Equippable with Proteinogenic or Taggable/Linkable Side Chains, General Promoters of Unusual Secondary Structures, «JOURNAL OF ORGANIC CHEMISTRY», 2019, 84, pp. 4992 - 5004 [articolo]
Baiula, M; Spampinato, S; Gentilucci, L ; Tolomelli, A, Novel Ligands Targeting alpha(4)beta(1) Integrin: Therapeutic Applications and Perspectives, «FRONTIERS IN CHEMISTRY», 2019, 7, Article number: 489, pp. 1 - 12 [articolo]Open Access
De Marco, Rossella; Bedini, Andrea; Spampinato, Santi*; Comellini, Lorenzo; Zhao, Junwei; Artali, Roberto; Gentilucci, Luca, Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 5751 - 5757 [articolo]Open Access
Dattoli, Samantha Deianira; Baiula, Monica; De Marco, Rossella; Bedini, Andrea; Anselmi, Michele; Gentilucci, Luca; Spampinato, Santi*, DS-70, a novel and potent α4 integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs, «BRITISH JOURNAL OF PHARMACOLOGY», 2018, 175, pp. 3891 - 3910 [articolo]Open Access
De Marco, Rossella; Greco, Arianna; Calonghi, Natalia; Dattoli, Samantha D.; Baiula, Monica; Spampinato, Santi; Picchetti, Pierre; De Cola, Luisa; Anselmi, Michele; Cipriani, Francesca; Gentilucci, Luca*, Selective detection of alfa4beta1 integrin (VLA-4)-expressing cells using peptide-functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites, «PEPTIDE SCIENCE», 2018, 110, Article number: e23081, pp. 1 - 10 [articolo]
Adamska-Bartłomiejczyk, Anna; De Marco, Rossella; Gentilucci, Luca; Kluczyk, Alicja; Janecka, Anna, Design and characterization of opioid ligands based on cycle-in-macrocycle scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY», 2017, 25, pp. 2399 - 2405 [articolo]