Uliassi, Elisa*; Prati, Federica; Bongarzone, Salvatore; Bolognesi, Maria Laura, Medicinal Chemistry of Hybrids for Neurodegenerative Diseases, in: Uliassi, Elisa*, Design of Hybrid Molecules for Drug Development, oxford, Elsevier Inc., 2017, pp. 259 - 277 [Chapter or essay]
Bruno, Stefano; Uliassi, Elisa; Zaffagnini, Mirko; Prati, Federica; Bergamini, Christian; Amorati, Riccardo; Paredi, Gianluca; Margiotta, Marilena; Conti, Paola; Costi, Maria Paola; Kaiser, Marcel; Cavalli, Andrea; Fato, Romana; Bolognesi, Maria Laura, Molecular basis for covalent inhibition of glyceraldehyde-3-phosphate dehydrogenase by a 2-phenoxy-1,4-naphthoquinone small molecule, «CHEMICAL BIOLOGY & DRUG DESIGN», 2017, 89, pp. 1 - 11 [Scientific article]
Uliassi, Elisa; Gandini, Annachiara; Perone, Rosaria Carmela; Bolognesi, Maria Laura*, Neuroregeneration versus neurodegeneration: Toward a paradigm shift in Alzheimer's disease drug discovery, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 995 - 1013 [Scientific article]
Jeřábek, Jakub; Uliassi, Elisa; Guidotti, Laura; Korábečný, Jan; Soukup, Ondřej; Sepsova, Vendula; Hrabinova, Martina; Kuča, Kamil; Bartolini, Manuela; Peña-Altamira, Luis Emiliano; Petralla, Sabrina; Monti, Barbara; Roberti, Marinella; Bolognesi, Maria Laura, Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 127, pp. 250 - 262 [Scientific article]
Bolognesi, Maria Laura; Gandini, Annachiara; Prati, Federica; Uliassi, Elisa, From Companion Diagnostics to Theranostics: A New Avenue for Alzheimer's Disease?, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 7759 - 7770 [Scientific article]
Junker, Anna; Balasubramanian, Ramachandran; Ciancetta, Antonella; Uliassi, Elisa; Kiselev, Evgeny; Martiriggiano, Chiara; Trujillo, Kevin; Mtchedlidze, Giorgi; Birdwell, Leah; Brown, Kyle A.; Harden, T. Kendall; Jacobson, Kenneth A, Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 6149 - 6168 [Scientific article]
Patent n. PCT Application No. PCT/US2016/053397, TRIAZOLE DERIVATIVES AS P2Y14 RECEPTOR ANTAGONISTS.
Patent n. US10683277B2, Triazole derivatives as P2Y14 receptor antagonists.
Kiselev, Evgeny; Balasubramanian, Ramachandran; Uliassi, Elisa; Brown, Kyle A.; Trujillo, Kevin; Katritch, Vsevolod; Hammes, Eva; Stevens, Raymond C.; Harden, T. Kendall; Jacobson, Kenneth A., Design, synthesis, pharmacological characterization of a fluorescent agonist of the P2Y14 receptor, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 4733 - 4739 [Scientific article]
Santucci, Matteo; Vignudelli, Tatiana; Ferrari, Stefania; Mor, Marco; Scalvini, Laura; Bolognesi, Maria Laura; Uliassi, Elisa; Costi, Maria Paola, The Hippo Pathway and YAP/TAZ-TEAD Protein-Protein Interaction as Targets for Regenerative Medicine and Cancer Treatment, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 4857 - 4873 [Scientific article]
Patent n. U.S. Patent Application No. 62/233,162, TRIAZOLE DERIVATIVES AS P2Y14 RECEPTOR ANTAGONISTS.
Eugenie Nepovimova;Elisa Uliassi;Jan Korabecny;Luis Emiliano Peña-Altamira;Sarah Samez;Alessandro Pesaresi;Gregory E. Garcia;Manuela Bartolini;Vincenza Andrisano;Christian Bergamini;Romana Fato;Doriano Lamba;Marinella Roberti;Kamil Kuca;Barbara Monti;Maria Laura Bolognesi, Multitarget Drug Design Strategy: Quinone–Tacrine Hybrids Designed To Block Amyloid-β Aggregation and To Exert Anticholinesterase and Antioxidant Effects, «JOURNAL OF MEDICINAL CHEMISTRY», 2014, 57, pp. 8576 - 8589 [Scientific article]
Federica Belluti;Elisa Uliassi;Giacomo Veronesi;Christian Bergamini;Marcel Kaiser;Reto Brun;Angelo Viola;Romana Fato;Paul A. M. Michels;R. Luise Krauth-Siegel;Andrea Cavalli;Maria Laura Bolognesi, Toward the Development of Dual-Targeted Glyceraldehyde-3-phosphate Dehydrogenase/Trypanothione Reductase Inhibitors againstTrypanosoma bruceiandTrypanosoma cruzi, «CHEMMEDCHEM», 2014, 9, pp. 371 - 382 [Scientific article]
F. Prati;E. Uliassi;M. L. Bolognesi, Two diseases, one approach: multitarget drug discovery in Alzheimer's and neglected tropical diseases, «MEDCHEMCOMM», 2014, 5, pp. 853 - 861 [Scientific article]